Permeability assay (Caco-2, MDCK, MDR1-MDCK etc.)

Plasma Protein Binding

Metabolic stability (Blood, Plasma, Microsomes, S9, Hepatocyte)

Drug-drug interaction:

CYP450 inhibition

CYP450 induction

CYP450 phenotype

Transporter (P-gp, BCRP, OATP, OCT, etc.)

Met ID

Blood Plasma Ratio